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  2. Discovery and development of HIV-protease inhibitors

    en.wikipedia.org/wiki/Discovery_and_development...

    Protease inhibitors can alter adipocyte metabolism causing lipodystrophy, a common side effect associated with the use of most HIV protease inhibitors. Many mechanisms have been proposed, for example inhibition of adipocyte differentiation, triglyceride accumulation and increased lipolysis. Theories considering the effect of protease inhibitors ...

  3. Protease inhibitor (pharmacology) - Wikipedia

    en.wikipedia.org/wiki/Protease_inhibitor...

    These protease inhibitors prevent viral replication by selectively binding to viral proteases (e.g. HIV-1 protease) and blocking proteolytic cleavage of protein precursors that are necessary for the production of infectious viral particles. Protease inhibitors that have been developed and are currently used in clinical practice include:

  4. HIV-1 protease - Wikipedia

    en.wikipedia.org/wiki/HIV-1_protease

    HIV-1 protease or PR is a ... In a general aspartic protease mechanism, once the substrate is properly bound to the active site of the enzyme, the deprotonated Asp25 ...

  5. Saquinavir - Wikipedia

    en.wikipedia.org/wiki/Saquinavir

    Saquinavir is a protease inhibitor. Proteases are enzymes that cleave protein molecules into smaller fragments. HIV protease is vital for both viral replication within the cell and release of mature viral particles from an infected cell.

  6. Aspartic protease - Wikipedia

    en.wikipedia.org/wiki/Aspartic_protease

    Proposed mechanism of peptide cleavage by aspartyl proteases. [6] Aspartyl proteases are a highly specific family of proteases – they tend to cleave dipeptide bonds that have hydrophobic residues as well as a beta-methylene group. Unlike serine or cysteine proteases these proteases do not form a covalent intermediate during cleavage ...

  7. Nelfinavir - Wikipedia

    en.wikipedia.org/wiki/Nelfinavir

    Nelfinavir is a protease inhibitor: it inhibits HIV-1 and HIV-2 proteases. HIV protease is an aspartate protease which splits viral protein molecules into smaller fragments, and it is vital to both the replication of the virus within the cell, and also to the release of mature viral particles from an infected cell.

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