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  2. GABA receptor agonist - Wikipedia

    en.wikipedia.org/wiki/GABA_receptor_agonist

    Gamma-aminobutyric acid, a GABA-B receptor agonist. A GABA receptor agonist is a drug that is an agonist for one or more of the GABA receptors, producing typically sedative effects, and may also cause other effects such as anxiolytic, anticonvulsant, and muscle relaxant effects. [1] There are three receptors of the gamma-aminobutyric acid. The ...

  3. Category:GABAA receptor agonists - Wikipedia

    en.wikipedia.org/wiki/Category:GABAA_receptor...

    Pages in category "GABA A receptor agonists" The following 20 pages are in this category, out of 20 total. This list may not reflect recent changes. A.

  4. GABA receptor - Wikipedia

    en.wikipedia.org/wiki/GABA_receptor

    The GABA receptors are a class of receptors that respond to the neurotransmitter gamma-aminobutyric acid (GABA), the chief inhibitory compound in the mature vertebrate central nervous system. There are two classes of GABA receptors: GABA A and GABA B .

  5. GABAA receptor - Wikipedia

    en.wikipedia.org/wiki/GABAA_receptor

    The ionotropic GABA A receptor protein complex is also the molecular target of the benzodiazepine class of tranquilizer drugs. Benzodiazepines do not bind to the same receptor site on the protein complex as does the endogenous ligand GABA (whose binding site is located between α- and β-subunits), but bind to distinct benzodiazepine binding sites situated at the interface between the α- and ...

  6. GABAA receptor positive allosteric modulator - Wikipedia

    en.wikipedia.org/wiki/GABAA_receptor_positive...

    However, they have no effect if GABA or another agonist is not present. Unlike GABA A receptor agonists, GABA A PAMs do not bind at the same active site as the γ-aminobutyric acid (GABA) neurotransmitter molecule: they affect the receptor by binding at a different site on the protein. This is called allosteric modulation. In psychopharmacology ...

  7. List of benzodiazepines - Wikipedia

    en.wikipedia.org/wiki/List_of_benzodiazepines

    IC 50 / pIC 50 values represent binding affinity only and do not reflect efficacy or pharmacokinetics, and some compounds listed are GABA A antagonists rather than agonists (e.g. flumazenil). Low IC 50 or high pIC 50 values indicate tighter binding (pIC 50 of 8.0 = IC 50 of 10nM, pIC 50 of 9.0 = IC 50 of 1nM, etc.)

  8. GABA analogue - Wikipedia

    en.wikipedia.org/wiki/GABA_analogue

    A GABA analogue is a compound which is an analogue or derivative of the neurotransmitter gamma-Aminobutyric acid (GABA) (the IUPAC of which is 4-aminobutanoic acid). Many GABA analogues are used as drugs , especially as anticonvulsants , sedatives , and anxiolytics .

  9. List of investigational sleep drugs - Wikipedia

    en.wikipedia.org/wiki/List_of_investigational...

    This is a list of investigational sleep drugs, ... EVT-201 – GABA A receptor positive allosteric ... – OX 2 receptor agonist pill (orally available) [2 ...